Preparation of Azepinoindole Derivatives via Oxidative Palladium Couplings

Lionel Joucla; Cyril Montagne; Guy Fournet; Benoit Joseph

doi:10.2174/157017805774717490

ISSN: 1570-1786
E-ISSN: 1875-6255

Preparation of Azepinoindole Derivatives via Oxidative Palladium Couplings
Authors: Lionel Joucla¹, Cyril Montagne², Guy Fournet³ and Benoit Joseph⁴
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¹ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France. ² Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France. ³ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France. ⁴ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France.
Source: Letters in Organic Chemistry, Volume 2, Issue 8, Dec 2005, p. 707 - 711
DOI: https://doi.org/10.2174/157017805774717490
- Available online: 01 Dec 2005

Abstract

Oxidative palladium couplings allow the preparation in high yields of different azepinoindole moieties. The use of CuCl2 as reoxidant leads to the formation of chloro derivatives instead of alkenes.

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2005-12-01

2025-09-11

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Article Type: Review Article

Keyword(s): Indole; oxidant; oxidative cyclisation; palladium

Preparation of Azepinoindole Derivatives via Oxidative Palladium Couplings

Abstract

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