Synthesis of 14-Membered Ring Jaspamide Derivatives

S. Celanire; C. Descamps-Francois; B. Lesur; G. Guillaumet; B. Joseph

doi:10.2174/1570178054640697

ISSN: 1570-1786
E-ISSN: 1875-6255

Synthesis of 14-Membered Ring Jaspamide Derivatives
Authors: S. Celanire¹, C. Descamps-Francois², B. Lesur³, G. Guillaumet⁴ and B. Joseph⁵
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¹ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France; ² Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France; ³ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France; ⁴ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France; ⁵ Laboratoire de Chimie Organique 1, UMR - CNRS 5181, Universite Claude Bernard - Lyon 1, CPE - Batiment 308, 43 Boulevard du 11 Novembre 1918, 69622 Villeurbanne Cedex, France;
Source: Letters in Organic Chemistry, Volume 2, Issue 6, Sep 2005, p. 528 - 531
DOI: https://doi.org/10.2174/1570178054640697
- Available online: 01 Sep 2005

Abstract

Two synthetic approaches of simpler jaspamide derivatives were investigated. The ring closure step was attempted either by RCM or by macrolactonisation. 14-Membered ring derivatives 15-16 were prepared by final macrolactonisation using Yamaguchi reagent.

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2005-09-01

2025-09-03

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Article Type: Review Article

Keyword(s): alkaloid; macrocycle; macrolactonisation; olefin metathesis

Synthesis of 14-Membered Ring Jaspamide Derivatives

Abstract

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