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- ISSN: 0929-8665
- E-ISSN: 1875-5305
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Synthesis of Alkyl and Aryl Esters of N-Protected β-Homoamino Acids from N-Protected α-Aminodiazoketones
- Source: Protein and Peptide Letters, Volume 9, Issue 6, Dec 2002, p. 529 - 532
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- 01 Dec 2002
Abstract
A simple and concomitant esterification method for the synthesis of methyl, ethyl, t-butyl, benzyl, and 9-fluorenylmethyl esters of Fmoc- / Boc- / Z-β-homoamino acids employing Fmoc- / Boc- / Z-α- aminodiazoketones by Wolff rearrangement is described. The method offers good yield with purity.
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