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Drug Metabolism Letters
In vitro systems including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics toxicokinetics species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; recent developments for the identification of drug metabolites reactive intermediate and glutathione conjugates.
Drug Metabolism and Bioanalysis
The scope includes in vitro systems including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics toxicokinetics species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; bioactivation; recent developments for the identification of drug metabolites reactive intermediate and glutathione conjugates.
Additionally LC/MS and other key detection methods including ligand binding assays sample preparation chromatography and separation sciences and method development and validation are included with applications in drug and metabolite assays pharmacokinetic/toxicokinetic assays biomarker assays immunogenicity assays diagnostic assays. Topics covered in this interdisciplinary journal include:
- Analytical Method and Drug Metabolism
- Bioavailability and Biopharmacy
- Cytochrome 450 Drug Metabolism
- Cytotoxicity
- Drug Absorption and Disposition
- Drug Biotransformation
- Drug Delivery System
- Drug-Drug Interaction
- Drug Food Interaction
- Drug Metabolizing Enzymes
- Drug Toxicology
- Drug Transporters
- Drugs and CYP2D6
- Factors Affecting Drug Metabolism
- Hepatic Metabolism of Drugs
- P-Glycoprotein and Transport Carriers
- Pharmacokinetics and Pharmacodynamics
- Phase I and II Drug Metabolism
- Reactive Metabolites
- Therapeutic Drug Monitoring
- Xenobiotics
Drug Metabolism and Bioanalysis Letters
Drug Metabolism and Bioanalysis Letters publishes letters original research articles mini-reviews thematic issues based on mini-reviews and letters commentaries technical notes and drug clinical trial studies on major advances in all areas of drug metabolism and bioanalysis.
In vitro systems including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics toxicokinetics species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; bioactivation; recent developments for the identification of drug metabolites reactive intermediate and glutathione conjugates. LC/MS and other key detection methods including ligand binding assays sample preparation chromatography and separation sciences method development and validation with applications in drug and metabolite assays pharmacokinetic/toxicokinetic assays biomarker assays immunogenicity assays diagnostic assays.